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Report error Found 4 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 2/G1/S-specific cyclin-E1' and Ligand = 'BDBM370326'
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM370326(BDBM467221 | US10233188, Example 213)
Affinity DataKi:  1.70nMAssay Description:Inhibition of recombinant full length wild-type phosphorylated CDK2/Cyclin E1 (unknown origin) expressed in baculovirus expression system assessed as...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM370326(BDBM467221 | US10233188, Example 213)
Affinity DataKi:  1.73nMAssay Description:The mobility shift assay electrophoretically separates the fluorescently labeled peptides (substrate and phosphorylated product) following the kinase...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent

TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM370326(BDBM467221 | US10233188, Example 213)
Affinity DataKi:  1.73nMAssay Description:The purpose of the CDK2/Cyclin E1 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a flu...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent

TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM370326(BDBM467221 | US10233188, Example 213)
Affinity DataKi:  1.73nMAssay Description:The purpose of the CDK2/Cyclin E1 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a flu...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent