Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 2' and Ligand = 'BDBM8037'
TargetCyclin-dependent kinase 2(Human)
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM8037(4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine...)
Affinity DataKi:  396nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM8037(4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine...)
Affinity DataIC50: 6.50E+3nMAssay Description:In vitro inhibition assay using human recombinant CDK2 and human recombinant cyclin A2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM8037(4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine...)
Affinity DataKd:  3.03E+4nMAssay Description:OctetRed_Method2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R

TargetCyclin-dependent kinase 2(Human)
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM8037(4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine...)
Affinity DataKon:  1.42M-1s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R

TargetCyclin-dependent kinase 2(Human)
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM8037(4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine...)
Affinity DataKoff:  8.22E+4s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R