Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Cysteinyl leukotriene receptor 1' and Ligand = 'BDBM50009070'
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50009070(CHEMBL22776 | 3-(2-Carboxy-ethylsulfanyl)-2-hydrox...)
Affinity DataKi:  5nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50009070(CHEMBL22776 | 3-(2-Carboxy-ethylsulfanyl)-2-hydrox...)
Affinity DataKi:  5nMAssay Description:Compound was evaluated for its ability to displace [3H]LTD4 from LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50009070(CHEMBL22776 | 3-(2-Carboxy-ethylsulfanyl)-2-hydrox...)
Affinity DataKi:  5nMAssay Description:Binding affinity against Cysteinyl leukotriene D4 receptor in guinea pig lung membranes using [3H]LTD4 as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50009070(CHEMBL22776 | 3-(2-Carboxy-ethylsulfanyl)-2-hydrox...)
Affinity DataKi:  10nMAssay Description:Binding affinity against Cysteinyl leukotriene D4 receptor in human lung membranes using [3H]LTD4 as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed