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Found 2 Enz. Inhib. hit(s) with Target = 'Cysteinyl leukotriene receptor 1' and Ligand = 'BDBM50084793'
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Laboratorios Menarini

Curated by ChEMBL
LigandPNGBDBM50084793(4-Oxo-2-(1H-tetrazol-5-yl)-4H-chromene-8-carboxyli...)
Affinity DataKi:  86nMAssay Description:In vitro binding affinity towards Cysteinyl leukotriene D4 receptor by using [3H]-LTD4 binding assay in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50084793(4-Oxo-2-(1H-tetrazol-5-yl)-4H-chromene-8-carboxyli...)
Affinity DataIC50:  86nMAssay Description:Antagonist activity at CysLT1 receptor in human dU937 cells assessed as inhibition of LTD4-induced increase of calcium level treated 30 mins before L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed