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Found 2 Enz. Inhib. hit(s) with Target = 'Cysteinyl leukotriene receptor 1' and Ligand = 'BDBM50084814'
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Laboratorios Menarini

Curated by ChEMBL
LigandPNGBDBM50084814(4-(4-(7-(quinolin-2-ylmethoxy)-2-naphthamido)pheny...)
Affinity DataKi:  1.5nMAssay Description:In vitro binding affinity towards Cysteinyl leukotriene D4 receptor by using [3H]-LTD4 binding assay in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50084814(4-(4-(7-(quinolin-2-ylmethoxy)-2-naphthamido)pheny...)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at CysLT1 receptor in human dU937 cells assessed as inhibition of LTD4-induced increase of calcium level treated 30 mins before L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed