Affinity DataKi: 1.00E+3nMAssay Description:Time dependent inhibition of CYP3A4-mediated testosterone-6-beta hydroxylation in human liver microsomeMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibition of human cytochrome P450 3A4More data for this Ligand-Target Pair