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Found 3 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 3A4' and Ligand = 'BDBM8885'
TargetCytochrome P450 3A4(Homo sapiens (Human))
Yanbian University College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM8885((1S,2R,10R,11S,14S,15S)-14-hydroxy-2,15-dimethylte...)
Affinity DataIC50:  45nMAssay Description:Inhibition of CYP3A4T (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetCytochrome P450 3A4(Homo sapiens (Human))
Yanbian University College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM8885((1S,2R,10R,11S,14S,15S)-14-hydroxy-2,15-dimethylte...)
Affinity DataIC50:  47nMAssay Description:Inhibition of CYP3A4T in human liver microsomes incubated for 15 to 40 mins in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetCytochrome P450 3A4(Homo sapiens (Human))
Yanbian University College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM8885((1S,2R,10R,11S,14S,15S)-14-hydroxy-2,15-dimethylte...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity for Cytochrome P450 3A4; Range = 1-10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank