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Found 2 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 3A5' and Ligand = 'BDBM50081468'
TargetCytochrome P450 3A5(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50081468(CHEMBL3422028)
Affinity DataKi:  855nMAssay Description:Inhibition of human recombinant CYP3A5 assessed as metabolism of 7-benzyloxy-4-trifluoromethylcoumarin to HFC after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A5(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50081468(CHEMBL3422028)
Affinity DataIC50:  556nMAssay Description:Inhibition of human recombinant CYP3A5 assessed as metabolism of 7-benzyloxy-4-trifluoromethylcoumarin to HFC after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed