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Found 3 Enz. Inhib. hit(s) with Target = 'D(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor' and Ligand = 'BDBM50327107'
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50327107((R)-methyl 2-(naphthalen-2-yl)-2-((R)-piperidin-2-...)
Affinity DataIC50:  33.9nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50327107((R)-methyl 2-(naphthalen-2-yl)-2-((R)-piperidin-2-...)
Affinity DataIC50:  34nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50327107((R)-methyl 2-(naphthalen-2-yl)-2-((R)-piperidin-2-...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity against dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed