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Found 2 Enz. Inhib. hit(s) with Target = 'D(1A) dopamine receptor' and Ligand = 'BDBM435987'
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM435987(2-(2,6-difluorophenyl)-1- ((1S,3R)-3-(hydroxymethy...)
Affinity DataEC50:  127nMAssay Description:Positive allosteric modulation of human D1 receptor expressed in HEK293 assessed as cAMP production incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM435987(2-(2,6-difluorophenyl)-1- ((1S,3R)-3-(hydroxymethy...)
Affinity DataEC50:  127nMAssay Description:The PAM activity of the compounds of the present invention may be measured essentially as described in Svensson et al., An Allosteric Potentiator of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent