Affinity DataKi: 1nMAssay Description:Binding affinity to dopamine D1 receptor high binding site by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity at rat striatal Dopamine receptor D1 using [3H]- SCH-23390 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Compound was evaluated for its ability to inhibit dopamine receptor D1 in rat striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Binding affinity to dopamine D1 receptor low binding site by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 730nMAssay Description:Displacement of [3H]SCH-23390 from rat dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+3nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:Binding affinity against Dopamine receptor D1 from rat brain corpus striatum membraneMore data for this Ligand-Target Pair
Affinity DataEC50: 1.86E+3nMAssay Description:Agonist activity at C-terminal RLuc8-fused D1R (unknown origin) transfected in human HEK293T cells co-expressing N-terminal Venus-tagged beta-arresti...More data for this Ligand-Target Pair
Affinity DataKd: 1.82E+3nMAssay Description:Equilibrium dissociation constant against recombinant Dopamine receptor D1A expressed in COS7 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.88E+3nMAssay Description:Agonist activity at C-terminal RLuc8-fused D1R (unknown origin) transfected in human HEK293T cells co-expressing N-terminal Venus-tagged beta-arresti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at D1R (unknown origin) transfected in human HEK293T cells assessed as increase in cAMP accumulation incubated for 2 hrs by cAMP Glo...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at D1R (unknown origin) transfected in human HEK293T cells assessed as increase in cAMP accumulation incubated for 2 hrs by cAMP Glo...More data for this Ligand-Target Pair