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Found 3 Enz. Inhib. hit(s) with Target = 'D(1A) dopamine receptor' and Ligand = 'BDBM50196234'
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50196234(8-methyl-5,6,7,8,9,10,15,16-octahydroindolo[3,2-g]...)
Affinity DataKi:  2.04nMAssay Description:Displacement of [3H]SCH23390 from human cloned dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50196234(8-methyl-5,6,7,8,9,10,15,16-octahydroindolo[3,2-g]...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]SCH 23390 from human D1 dopamine receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50196234(8-methyl-5,6,7,8,9,10,15,16-octahydroindolo[3,2-g]...)
Affinity DataKi:  2.80nMAssay Description:Activity at human D1 dopamine receptor expressed in HEK293 cells by calcium fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed