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Found 7 Enz. Inhib. hit(s) with Target = 'D(1B) dopamine receptor' and Ligand = 'BDBM50180913'
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to D5 dopamine receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human cloned dopamine D5 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  1.69nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  1.69nMAssay Description:Inhibition of D5 dopamine receptor in HEK 293 cells by intracellular calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed