TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: >1.00E+4nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Texas
Curated by PDSP Ki Database
University of North Texas
Curated by PDSP Ki Database
Affinity DataKi: 1.29E+4nMAssay Description:Inhibitory constant against binding of [125I]- IBZM to D2 receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: <5.01E+3nMAssay Description:Antagonist activity at human wild-type D2 receptor expressed in CHO-K1 cells assessed as dopamine-induced cAMP by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: <5.01E+3nMAssay Description:Agonist activity at human wild-type D2 receptor expressed in CHO-K1 cells assessed as cAMP level by HTRF assayMore data for this Ligand-Target Pair