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Found 3 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50052563'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50052563(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-(5-metho...)
Affinity DataKi:  253nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50052563(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-(5-metho...)
Affinity DataIC50:  761nMAssay Description:Binding affinity against Dopamine receptor D2 in rat striatal membrane using [3H]spiroperidol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50052563(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-(5-metho...)
Affinity DataIC50:  761nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed