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Found 3 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50066910'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita' Di Siena

Curated by ChEMBL
LigandPNGBDBM50066910((+/-)7-Chloro-9-(4-methyl-piperazin-1-yl)-9,10-dih...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]spiperone (Dopamine receptor D2) binding to rat tissue homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita' Di Siena

Curated by ChEMBL
LigandPNGBDBM50066910((+/-)7-Chloro-9-(4-methyl-piperazin-1-yl)-9,10-dih...)
Affinity DataKi:  3.80nMAssay Description:Half-maximal inhibition of [3H]spiperone binding to Dopamine receptor D2 in rat striatal homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita' Di Siena

Curated by ChEMBL
LigandPNGBDBM50066910((+/-)7-Chloro-9-(4-methyl-piperazin-1-yl)-9,10-dih...)
Affinity DataKi:  49.6nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]spiperone (Dopamine receptor D2) binding to rat tissue homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed