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Found 3 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50516522'
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516522(CHEMBL4447416)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516522(CHEMBL4447416)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516522(CHEMBL4447416)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cells measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed