Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with Target = 'D(3) dopamine receptor' and Ligand = 'BDBM50172506'
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172506(CHEMBL193337 | Dipropyl-(S)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  4nMAssay Description:High binding affinity towards human dopamine receptor 3 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172506(CHEMBL193337 | Dipropyl-(S)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  8.40nMAssay Description:Ligand efficacy towards dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172506(CHEMBL193337 | Dipropyl-(S)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]7-OH-DPAT from human dopamine D3 receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172506(CHEMBL193337 | Dipropyl-(S)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172506(CHEMBL193337 | Dipropyl-(S)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  110nMAssay Description:Low binding affinity towards human dopamine receptor 3 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172506(CHEMBL193337 | Dipropyl-(S)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]spiperone from wild type human dopamine D3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172506(CHEMBL193337 | Dipropyl-(S)-4,5,6,7-tetrahydro-pyr...)
Affinity DataEC50:  3.40nMAssay Description:Effective concentration against dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed