Affinity DataKi: 380nMAssay Description:Displacement of [3H]N-methylspiperone from human D3R receptor expressed in HEK293T cell membrane incubated for 1 hr by MicroBeta scintillation counti...More data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Ability to displace [3H]-spiperone from cloned human dopamine D3 receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Binding affinity towards cloned human Dopamine receptor D3 stably expressed in CHO cells was evaluated using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.31E+3nMAssay Description:Binding affinity to D3R (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.31E+3nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.03E+3nMAssay Description:Binding affinity at Dopamine receptor D3 in CHO cells by radioligand displacement.More data for this Ligand-Target Pair
Affinity DataKi: >3.03E+3nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity to cloned rat Dopamine receptor D3 measured by displacement of the radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+4nMAssay Description:Displacement of [3H]spiroperidol from human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+4nMAssay Description:In vitro binding affinity at human cloned dopamine receptor D3 stably expressed in CHO cells by [3H]spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.90E+4nMAssay Description:Binding affinity evaluated for the displacement of [3H]-spiperone against human dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 6.50E+4nMAssay Description:Displacement of [3H] Spiperone from human D3 receptor expressed in CHO cells by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Binding affinity to cloned human Dopamine receptor D3 expressed in CHO cells by [3H]spiperone displacement.More data for this Ligand-Target Pair