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Found 2 Enz. Inhib. hit(s) with Target = 'DNA gyrase subunit B' and Ligand = 'BDBM50330294'
TargetDNA gyrase subunit B(Escherichia coli (strain K12))
UniversitäT TüBingen

Curated by ChEMBL
LigandPNGBDBM50330294((2R,3R,4R,5R)-2-(3-(4-amino-3-methylbenzamido)-4-h...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Escherichia coli JM109 DNA gyrase subunit B assessed as DNA triple helix formation by supercoiling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Escherichia coli (strain K12))
UniversitäT TüBingen

Curated by ChEMBL
LigandPNGBDBM50330294((2R,3R,4R,5R)-2-(3-(4-amino-3-methylbenzamido)-4-h...)
Affinity DataIC50:  784nMAssay Description:Inhibition of Escherichia coli JM109 DNA gyrase subunit B assessed as ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed