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Found 4 Enz. Inhib. hit(s) with Target = 'DNA-dependent protein kinase catalytic subunit' and Ligand = 'BDBM50159678'
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50159678(3-Morpholin-4-yl-benzo[f]chromen-1-one | 3-morphol...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50159678(3-Morpholin-4-yl-benzo[f]chromen-1-one | 3-morphol...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of DNA dependent protein kinase isolated from HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50159678(3-Morpholin-4-yl-benzo[f]chromen-1-one | 3-morphol...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50159678(3-Morpholin-4-yl-benzo[f]chromen-1-one | 3-morphol...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against DNA-dependent protein kinase receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed