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Found 4 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM21021'
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Arizona Tucson

LigandPNGBDBM21021(Bifunctional Peptide Ligand, 5 (TY005) | CHEMBL389...)
Affinity DataKi:  2.80nM ΔG°:  -48.8kJ/mole EC50:  2.90nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Arizona Tucson

LigandPNGBDBM21021(Bifunctional Peptide Ligand, 5 (TY005) | CHEMBL389...)
Affinity DataIC50:  6.30nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cell membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21021(Bifunctional Peptide Ligand, 5 (TY005) | CHEMBL389...)
Affinity DataIC50:  22nMAssay Description:Agonist activity at delta opioid receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Arizona Tucson

LigandPNGBDBM21021(Bifunctional Peptide Ligand, 5 (TY005) | CHEMBL389...)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at human delta opioid receptor expressed in mouse HN9.10 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed