Affinity DataKi: 69nMAssay Description:Tested for inhibition of amplification of electrically induced twitch in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataKi: 69.1nMAssay Description:Binding affinity was determined on delta [3H]-DPDPE site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Tested for inhibition of amplification of electrically induced twitch in guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Binding affinity was determined on delta [3H]-DPDPE site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair