Affinity DataKi: 180nMAssay Description:Displacement of [3H]-DPN from rat DOR expressed in EE-HEK293 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+5nMAssay Description:Agonist activity at DOR in CD1 mouse vas deferens assessed as inhibition of EFS-induced contractions incubated for 60 minsMore data for this Ligand-Target Pair