Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM50334988'
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50334988((S)-2-amino-N-((R)-1-(2-((S)-3-(4-fluorophenyl)-1-...)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50334988((S)-2-amino-N-((R)-1-(2-((S)-3-(4-fluorophenyl)-1-...)
Affinity DataIC50:  1.80nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50334988((S)-2-amino-N-((R)-1-(2-((S)-3-(4-fluorophenyl)-1-...)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed