Affinity DataKi: 6.10nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Activity was evaluated in human delta opioid receptors transfected with CHO cells by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair