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Found 4 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 4' and Ligand = 'BDBM50171556'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataIC50:  0.890nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataIC50:  3.5nMpH: 2.0Assay Description:The inhibitor solution is prepared by dissolving 3-5 mg of inhibitor in pH 2 solution (0.01 N HCl), such that the concentration of the solution is eq...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataIC50:  9nMpH: 8.0Assay Description:The inhibitor solution is prepared by dissolving 3-5 mg of inhibitor in pH 2 solution (0.01 N HCl), such that the concentration of the solution is eq...More data for this Ligand-Target Pair
In DepthDetails US Patent