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Found 4 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 4' and Ligand = 'BDBM50206043'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206043(((2S,4S)-4-(4-(5-nitropyridin-2-yl)piperazin-1-yl)...)
Affinity DataIC50:  0.920nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206043(((2S,4S)-4-(4-(5-nitropyridin-2-yl)piperazin-1-yl)...)
Affinity DataIC50:  0.920nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206043(((2S,4S)-4-(4-(5-nitropyridin-2-yl)piperazin-1-yl)...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206043(((2S,4S)-4-(4-(5-nitropyridin-2-yl)piperazin-1-yl)...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed