Found 5 Enz. Inhib. hit(s) with Target = 'Dual serine/threonine and tyrosine protein kinase' and Ligand = 'BDBM2579'
TargetDual serine/threonine and tyrosine protein kinase(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 31.3nMAssay Description:Inhibition of human RIPK5 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetDual serine/threonine and tyrosine protein kinase(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 65.2nMAssay Description:Inhibition of human RIPK5 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetDual serine/threonine and tyrosine protein kinase(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of human RIPK5 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetDual serine/threonine and tyrosine protein kinase(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of human RIPK5 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetDual serine/threonine and tyrosine protein kinase(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Binding constant for RIPK5 kinase domainMore data for this Ligand-Target Pair