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Found 2 Enz. Inhib. hit(s) with Target = 'Dual specificity mitogen-activated protein kinase kinase 1/2' and Ligand = 'BDBM50209763'
TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50209763(CHEMBL3883792)
Affinity DataIC50:  400nMAssay Description:Inhibition of MEK1/2 in human HT-29 cells assessed as reduction in cell proliferation after 72 hrs by CellTiter-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50209763(CHEMBL3883792)
Affinity DataIC50:  400nMAssay Description:Inhibition of MEK1/2 in human HT-29 cells assessed as reduction in cell proliferation after 72 hrs by CellTiter-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed