Found 1 Enz. Inhib. hit(s) with Target = 'Dual specificity mitogen-activated protein kinase kinase 1' and Ligand = 'BDBM50391643'
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of N-terminal GST-tagged MEK1 after 5 mins by scintillation counterMore data for this Ligand-Target Pair