Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Dual specificity mitogen-activated protein kinase kinase 1 [2-31,52-393,S218E,S222D]' and Ligand = 'BDBM50337928'
TargetDual specificity mitogen-activated protein kinase kinase 1 [2-31,52-393,S218E,S222D](Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM50337928((R)-3-(2,3-dihydroxypropyl)-5-(4-ethynyl-2-fluorop...)
Affinity DataIC50: <5nMpH: 7.3 T: 2°CAssay Description:Reaction product is determined quantitatively by fluorescent polarization using progressive IMAP beads from Molecular Devices.More data for this Ligand-Target Pair
In DepthDetails US Patent