Found 5 Enz. Inhib. hit(s) with Target = 'Dual specificity protein kinase CLK1' and Ligand = 'BDBM50435473' TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human CLK1 (130 to end residues) using ERMRPRKRQGSVRRRV as substrate incubated for 40 mins in presence of [gamma33P-ATP] by...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human CLK1 expressed in Sf9 insect cells using myelin basic protein as substrate incubated for 110 mins in presence of ATP ...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human CLK1 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scinti...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant CLK1 (148 to 484 amino acids) expressed in Escherichia coli BL21(DE3) using AFRREWSPGKEAKK as substrate preincubated ...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataKd: 2.80nMAssay Description:Binding affinity to human CLK1 assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
