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Found 4 Enz. Inhib. hit(s) with Target = 'Dual specificity protein kinase CLK4' and Ligand = 'BDBM50326053'
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of recombinant human CLK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scinti...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd:  410nMAssay Description:Binding constant for CLK4 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd:  410nMAssay Description:Binding affinity to CLK4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd:  410nMAssay Description:Binding constant for CLK4 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed