Found 10 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1A' and Ligand = 'BDBM50070942' TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Avanti Biosciences
Curated by ChEMBL
Avanti Biosciences
Curated by ChEMBL
Affinity DataIC50: 232nMAssay Description:Inhibition of DYRK1A (unknown origin) using HT-497 as substrate preincubated with compound followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Avanti Biosciences
Curated by ChEMBL
Avanti Biosciences
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of human GST-fused DYRK1A expressed in Escherichia coli using KISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 330nMAssay Description:Inhibition of rat Dyrk1A using Woodtide as substrate after 40 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Avanti Biosciences
Curated by ChEMBL
Avanti Biosciences
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of human recombinant GST-tagged DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 40 mins in presence of [gamma...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Avanti Biosciences
Curated by ChEMBL
Avanti Biosciences
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Avanti Biosciences
Curated by ChEMBL
Avanti Biosciences
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Avanti Biosciences
Curated by ChEMBL
Avanti Biosciences
Curated by ChEMBL
Affinity DataIC50: 491nMAssay Description:Inhibition of recombinant human DYRK1A expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scin...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Avanti Biosciences
Curated by ChEMBL
Avanti Biosciences
Curated by ChEMBL
Affinity DataIC50: 766nMAssay Description:Inhibition of recombinant human DYRK1A expressed in Escherichia coli using DYRKtide peptide as substrate incubated for 110 mins in presence of ATP by...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Avanti Biosciences
Curated by ChEMBL
Avanti Biosciences
Curated by ChEMBL
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of GST-tagged human DYRK1A using dephosphorylated MBP as substrate after 10 mins by Kinase-Glo plus luminescent kinase assayMore data for this Ligand-Target Pair
