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Found 2 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1A' and Ligand = 'BDBM50341228'
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50341228(1-(4-fluoro-2-(trifluoromethyl)phenyl)-9-(1H-pyraz...)
Affinity DataKi:  252nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50341228(1-(4-fluoro-2-(trifluoromethyl)phenyl)-9-(1H-pyraz...)
Affinity DataIC50:  532nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair