Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1A' and Ligand = 'BDBM50445229'
LigandPNGBDBM50445229(CHEMBL3102953)
Affinity DataKi:  7.60nMAssay Description:Competitive inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using ATP as subst...More data for this Ligand-Target Pair
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LigandPNGBDBM50445229(CHEMBL3102953)
Affinity DataIC50:  14nMAssay Description:Inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using N-terminal fluorescein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed