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Found 2 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 4' and Ligand = 'BDBM50292406'
LigandPNGBDBM50292406(CHEMBL485053 | leucettamine B)
Affinity DataIC50:  6.37E+3nMAssay Description:Inhibition of recombinant human DYRK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scint...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50292406(CHEMBL485053 | leucettamine B)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged DYRK4 expressed in Escherichia coli using GRSRSRSRSRSR as substrate and [gamma33P]ATP after 30 mins by sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed