Found 3 Enz. Inhib. hit(s) with Target = 'E3 ubiquitin-protein ligase XIAP' and Ligand = 'BDBM50145767'
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of Michigan Comprehensive Cancer Center
Curated by ChEMBL
University Of Michigan Comprehensive Cancer Center
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Compound was tested for inhibiotry activity towards XIAP BIR3 proteinMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of Michigan Comprehensive Cancer Center
Curated by ChEMBL
University Of Michigan Comprehensive Cancer Center
Curated by ChEMBL
Affinity DataIC50: 2.83E+3nMAssay Description:Compound was tested for inhibiotry activity towards XIAP BIR3 proteinMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of Michigan Comprehensive Cancer Center
Curated by ChEMBL
University Of Michigan Comprehensive Cancer Center
Curated by ChEMBL
Affinity DataKd: 240nMAssay Description:Dissociation constant towards X-linked inhibitor of apoptosis (XIAP) BIR3 protein was determinedMore data for this Ligand-Target Pair