Found 2 Enz. Inhib. hit(s) with Target = 'E3 ubiquitin-protein ligase XIAP' and Ligand = 'BDBM50465628'
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 191nMAssay Description:Displacement of AVPIAQKSEK-biotin from N-terminal His-tagged human recombinant XIAP BIR3 (253 to 347 residues) expressed in Escherichia coli BL21(DE3...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataKd: 783nMAssay Description:Binding affinity to N-terminal His-tagged human recombinant XIAP BIR3 (253 to 347 residues) expressed in Escherichia coli BL21(DE3) Gold by isotherma...More data for this Ligand-Target Pair