Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'EEF1AKMT4-ECE2 readthrough transcript protein' and Ligand = 'BDBM50271179'
TargetEEF1AKMT4-ECE2 readthrough transcript protein(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

LigandPNGBDBM50271179(2-(2-(quinolin-2-yl)vinyl)phenol | CHEMBL487942 | ...)
Affinity DataIC50:  1.60E+3nMpH: 5.5Assay Description:Recombinant ECE2 (32.5 ng) with a specific activity of 12 pmol/min/μg protein was generated as described previously. Secreted soluble recombinan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEEF1AKMT4-ECE2 readthrough transcript protein(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

LigandPNGBDBM50271179(2-(2-(quinolin-2-yl)vinyl)phenol | CHEMBL487942 | ...)
Affinity DataIC50:  4.63E+3nMAssay Description:Reduction of recombinant ECE2 (unknown origin) activity measured by McaBk2 fluorescent substrate hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed