Found 4 Enz. Inhib. hit(s) with Target = 'Endoplasmic reticulum aminopeptidase 1' and Ligand = 'BDBM50519944' TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Kansas University Specialized Chemistry Center
Curated by ChEMBL
Kansas University Specialized Chemistry Center
Curated by ChEMBL
Affinity DataKi: 1.28E+4nMAssay Description:Competitive inhibition of recombinant human C-terminal His6-tagged ERAP1 expressed in baculovirus infected BTA-TN-5B1-4 insect cells using varying le...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Kansas University Specialized Chemistry Center
Curated by ChEMBL
Kansas University Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of recombinant human C-terminal His6-tagged ERAP1 expressed in baculovirus infected BTA-TN-5B1-4 insect cells using WRCYEKMALK as substrat...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Kansas University Specialized Chemistry Center
Curated by ChEMBL
Kansas University Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of recombinant human C-terminal His6-tagged ERAP1 expressed in baculovirus infected BTA-TN-5B1-4 insect cells using L-AMC as substrate mea...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Kansas University Specialized Chemistry Center
Curated by ChEMBL
Kansas University Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of ERAP1 in human HeLa cells stably expressing H-2 Kb infected with vaccinia virus containing ss-LEQLE-SIINFEKL epitope assessed as suppre...More data for this Ligand-Target Pair
