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Found 3 Enz. Inhib. hit(s) with Target = 'Endothelin receptor type B' and Ligand = 'BDBM50395633'
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50395633(CHEMBL2165332)
Affinity DataIC50:  441nMAssay Description:Displacement of [I125]ET1 from recombinant ETB receptor expressed in CHO cells after 2 hrs by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50395633(CHEMBL2165332)
Affinity DataIC50:  441nMAssay Description:Antagonist activity at ETB receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50395633(CHEMBL2165332)
Affinity DataIC50:  441nMAssay Description:Antagonist activity at ETB receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed