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Found 3 Enz. Inhib. hit(s) with Target = 'Endothelin-1 receptor' and Ligand = 'BDBM50000553'
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000553((S)-3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000553((S)-3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [125I]endothelin-1 [ET-1] binding to endothelin A receptor (ETA) of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000553((S)-3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50:  5.80E+4nMAssay Description:Compound was evaluated for the binding affinity to endothelin receptor in the rat heart ventricle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed