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Found 3 Enz. Inhib. hit(s) with Target = 'Endothelin-1 receptor' and Ligand = 'BDBM50056071'
TargetEndothelin-1 receptor(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50056071((2R,3R,4S)-4-Benzofuran-5-yl-1-dibutylcarbamoylmet...)
Affinity DataIC50:  0.480nMAssay Description:Binding affinity against endothelin A receptor in MMQ cells in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50056071((2R,3R,4S)-4-Benzofuran-5-yl-1-dibutylcarbamoylmet...)
Affinity DataIC50:  0.5nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50056071((2R,3R,4S)-4-Benzofuran-5-yl-1-dibutylcarbamoylmet...)
Affinity DataIC50:  0.5nMAssay Description:Binding affinity towards endothelin A receptor in prolactin secreting rat pituitary cells using [125I]-ET-1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed