Affinity DataIC50: 0.00620nMAssay Description:Ability to inhibit [125I]ET1 binding to endothelin A receptor in porcine aortic membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0150nMAssay Description:Displacement of 125I-ET1 from ETA receptor in rat A7R5 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0150nMAssay Description:Displacement of 125I-ET1 from ETA receptor in rat A7R5 cellsMore data for this Ligand-Target Pair
TargetEndothelin-1 receptor(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv)
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at ET-A receptor (unknown origin)More data for this Ligand-Target Pair
TargetEndothelin-1 receptor(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv)
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Displacement of [I125]ET1 from recombinant ETA receptor expressed in CHO cells after 2 hrs by TopCount analysisMore data for this Ligand-Target Pair