Found 1 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor [L858R,C797S]' and Ligand = 'BDBM50185140' TargetEpidermal growth factor receptor [L858R,C797S](Homo sapiens (Human))
Chengdu Di''Ao Jiuhong Pharmaceutical Factory
US Patent
Chengdu Di''Ao Jiuhong Pharmaceutical Factory
US Patent
Affinity DataIC50: 548nMAssay Description:To assess the effect of compounds on the activity of wild-type and mutant EGFR kinases, kinase activity was tested by measuring ATP consumption in an...More data for this Ligand-Target Pair
3D Structure (crystal)