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Found 1 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM22433'
TargetEstrogen receptor(Homo sapiens (Human))
Gsk

LigandPNGBDBM22433(4-hydroxytamoxifen (4-OHT) analog, 13 | N-[(4Z)-5-...)
Affinity DatapH: 7.4 T: 2°CAssay Description:Binding affinity was measured by a scintillation proximity binding assay using [3H]4-OHT (for ERRgamma) or [3H]estradiol (for ERalpha) as radioligand...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed