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Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM349617'
TargetEstrogen receptor(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM349617((3-(4-(2-(sec- butylamino)ethyl)phenoxy)-6- hydrox...)
Affinity DataIC50: <1.00E+3nMAssay Description:All reagents used in this assay was supplied in the Human ERα Reporter Assay by Indigo Biosciences #IB00401. In an effort to screen selective es...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM349617((3-(4-(2-(sec- butylamino)ethyl)phenoxy)-6- hydrox...)
Affinity DataIC50: <1.00E+3nMAssay Description:A screening strategy was implemented utilizing an In-Cell Western assay to measure their ability to degrade the estrogen receptor in vitro. MCF7 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent