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Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM368202'
TargetEstrogen receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM368202(US10227334, Example 2-(4-((S)-2-(azetidin-1-yl)pro...)
Affinity DataIC50:  0.900nMAssay Description:Induction of ERalpha degradation in human MCF7 cells in phenol red free RPMI medium containing 5% charcoal dextran-treated FBS incubated for 4 hrs by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM368202(US10227334, Example 2-(4-((S)-2-(azetidin-1-yl)pro...)
Affinity DataIC50:  100nMAssay Description:MCF-7 cells were adjusted to a concentration of 40,000 cells per mL in RPMI containing 10% FBS and 20 mM HEPES. 16 microliters of the cell suspension...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent